沈阳药科大学学报

2001, (01) 18-19

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马来酸罗格列酮的合成工艺改进
An improved synthesis of rosiglitazone maleate

付晔,王绍杰,张为革,许越
FU Ye; WANG Shao jie; ZHANG Wei ge; XU Yue (Department of Pharmaceutics;

摘要(Abstract):

对马来酸罗格列酮的合成方法进行改进 ,5步反应总收率为 2 8 6 %
Rosiglitazone maleate was synthesized through an improved method.The total yield was improved from 13 1% to 28 6%.

关键词(KeyWords): 抗糖尿病药;马来酸罗格列酮;合成
antidiabetic drug; rosiglitazone maleate; synthe?

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作者(Authors): 付晔,王绍杰,张为革,许越
FU Ye; WANG Shao jie; ZHANG Wei ge; XU Yue (Department of Pharmaceutics;

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